产品描述
Agomelatine对5-HT2C受体具有拮抗作用,因而是一种去甲肾上腺素-多巴胺***解除剂(NDDI)。Agomelatine is structurally closely related to melatonin. Agomelatine is a potent agonist at melatonin receptors and an antagonist at serotonin-2C (5-HT2C) receptors, tested in an animal model of depression.
产品价格
货号 | 规格 | 价格 |
CC1399 |
10mg |
670.00 元 |
CC1399 | 50mg | 1970.00 元 |
CC1399 | 100mg | 3170.00 元 |
CC1399 | 200mg | 4870.00 元 |
化学数据
分子量Molecular Weight (MW) | 243.3 | |
---|---|---|
化学式Formula |
C15H17NO2 |
|
CAS号CAS No. | 138112-76-2 | |
溶解性Solubility (25°C) | 二甲基亚砜DMSO | 48 mg/mL(197.28 mM) |
水Water | Insoluble | |
乙醇Alcohol | 48 mg/mL(197.28 mM) |
制备储备液
浓度/溶剂体积(DMSO)/质量 | 1 mg | 5 mg | 10 mg |
1 mM | 4.1102 mL | 20.5508 mL | 41.1015 mL |
5 mM | 0.8220 mL | 4.1102 mL | 8.2203 mL |
10 mM | 0.4110 mL | 2.0551 mL | 4.1102 mL |
50 mM | 0.0822 mL | 0.4110 mL | 0.8220 mL |